agent chemical name syn use/assay/comment
miscellaneous
urethane (ethyl carbamate)   *one of first organic cpd show anticancer activity*test of identity :hyd by acid or alkali *structure is very restrictive >any change abolish activity or less active
colchicine & demeclocine colchicine R=COCH3 , Demeclocine R=CH3 alkaloid isolated from plant colchicum autumnale *cholchicine :antimitotic ,demeclocine :myelocytic leukaemia **assay :alkaloidal assay
cisplatin (Platinol ,platinex) cis-dichlorodiammine platinum II *used in combination e bleomycin & Vinblastine ** used in testicular tumour
carboplatin (paraplatin) 1,1-cyclobutane dicarboxylic acid platinum diammine complex   *str related to cisplatin e reduced nephrotoxicity *used in ttt of ovarian carcinoma & lung cancer
Mitolactor (Dibromodulcitol) 1,6-dibromo galactitol or 1,6-dibromo dulcitol   mech of action :alkylating agent
Hydroxyurea (Hydrea ,hydroxycarbamide) hydroxycarbamide *mech :ribonucleotide reductase inhibitor ,inhibit DNA syn -*uses :melanoma ,chronic myelocytic leukemia ,inoperable carcinoma of ovary ,in combination of irradiation therapy for carcinomas of head & neck
Dacarbazine (Deticene) 5-(Dimethyltriazeno) imidazole-4-carboxamide  
Procarbazine HCl (Natulan) 4-(2-methyl hydrazinomethyl)-N-isopropyl benzamide  
Tamoxifen citrate  (Tamofen ,Nolvadex) 1-(p-B-dimethylamino ethoxy phenyl) trans-1,2diphenyl -but-1-ene used in ttt & prevention of breast cancer
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